The principles above are not abstractions; they were forged by, and are visible in, the small set of human trials that now define the field. The exemplar is TAME — Targeting Aging with Metformin — conceived explicitly as a regulatory proof of concept rather than a bet on a particular drug (Barzilai et al., 2016). Its design embodies every move of this chapter: metformin, a cheap and exhaustively characterised diabetes drug, tested in older adults against a composite of age-related outcomes — major cardiovascular events, cancer, dementia and death — with the supporting biomarker panel running underneath (Justice et al., 2018). The point was never that metformin is the ideal geroprotector; the meta-analytic evidence in animals is in fact stronger for rapamycin, which mirrors dietary restriction in a way metformin does not (Ivimey-Cook et al., 2025). The point was to establish that a trial against ageing can be designed, run and read — to cut the regulatory path that successors would walk.
Its complement is PEARL, a decentralised trial of low-dose rapamycin that reported acceptable safety and several healthspan signals over a year in a community of self-selected participants, demonstrating both the promise and the limits of the remote, participant-driven model (Moel et al., 2025). Beyond these, the wider landscape is consistent in a way this chapter has prepared us to expect: the first-in-human senolytic studies measured feasibility, tolerability and target engagement — that the drugs reach their tissues and lower senescent-cell burden — rather than disease outcomes (Section 7.3) (Hickson et al., 2019; Justice et al., 2019); the CALERIE analysis read biological age with clocks rather than counting deaths (Waziry et al., 2023); and the reprogramming therapies of Chapter 8 approach their first human tests with the dosing-and-endpoint problem of Section 8.2 still squarely before them. Table 10.1 sets the principal trials side by side.
The common thread is unmistakable. These are, almost to a trial, studies of whether the intervention does what its mechanism says — reaches the target, moves the marker, proves tolerable — and not yet studies of whether it lengthens a healthy life. That is the appropriate state of an early translational field, and nothing to apologise for. But it places an unusual burden on the reader of longevity science, who must constantly distinguish a moved biomarker from a changed destiny, and a regulable composite from a proven benefit.
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